A concise and scalable strategy for the total synthesis of dictyodendrin B based on sequential C-H functionalization.
نویسندگان
چکیده
A sequential CH functionalization strategy for the synthesis of the marine alkaloid dictyodendrin B is reported. Our synthesis begins from commercially available 4-bromoindole and involves six direct functionalizations around the heteroarene core as part of a gram-scale strategy towards the natural product.
منابع مشابه
Total synthesis of dictyodendrin B.
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ورودعنوان ژورنال:
- Angewandte Chemie
دوره 54 18 شماره
صفحات -
تاریخ انتشار 2015